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			{{cs1 config|name-list-style=vanc}}
	{{Chembox		{{Chembox
			| Verifiedfields = changed
			| Watchedfields = changed
			| verifiedrevid = 477238724
	| ImageFile = Acetarsol.svg		| ImageFile = Acetarsol.svg
		⚫	| ImageFile_Ref = {{chemboximage|correct|??}}
	| ImageSize = 244		| ImageSize = 244
	| ImageName = Structural formula of acetarsol		| ImageName = Kekulé, skeletal formula of acetarsol
	| PIN = Acetarsone
	| SystematicName = (3-Acetamido-4-hydroxyphenyl)arsonic acid		| PIN = (3-Acetamido-4-hydroxyphenyl)arsonic acid
	| OtherNames = 3-Acetamido-4-hydroxyphenylarsonic acid		| OtherNames = Acetarsone
	| Section1 = {{Chembox Identifiers		|Section1={{Chembox Identifiers
		⚫	| CASNo_Ref = {{cascite|correct|CAS}}
	| CASNo = 97-44-9		| CASNo = 97-44-9
⚫	| CASNo_Ref = {{cascite|correct|??}}
	| PubChem = 1985		| ChEBI = 135135
	| PubChem_Ref = {{Pubchemcite|correct|PubChem}}		| ChEMBL_Ref = {{ebicite|correct|EBI}}
			| ChEMBL = 1330792
⚫	| ChemSpiderID = 1908
			| DrugBank = DB13268
⚫	| ChemSpiderID_Ref = {{chemspidercite|correct|chemspider}}
	| UNII = 806529YU1N		| PubChem = 1985
		⚫	| ChemSpiderID = 1908
⚫	| UNII_Ref = {{fdacite|correct|FDA}}
		⚫	| ChemSpiderID_Ref = {{chemspidercite|correct|chemspider}}
⚫	| EINECS = 202-582-3
	| KEGG = D07110		| UNII = 806529YU1N
			| UNII_Ref = {{fdacite|correct|FDA}}
⚫	| MeSHName = Acetarsol
		⚫	| EINECS = 202-582-3
⚫	| ATCCode_prefix = A07
	| ATCCode_suffix = AX02		| UNNumber = 3465
			| KEGG_Ref = {{keggcite|correct|kegg}}
	| ATC_Supplemental = G01AB01, P01CD02, P51AD05
			| KEGG = D07110
	| SMILES = O=(O)(O)c1ccc(O)c(NC(=O)C)c1
		⚫	| MeSHName = Acetarsol
⚫	| SMILES1 = CC(=O)NC1=CC(=CC=C1O)(O)(O)=O
			| SMILES = CC(=O)Nc1cc(ccc1O)(O)(O)=O
⚫	| StdInChI = 1S/C8H10AsNO5/c1-5(11)10-7-4-6(9(13,14)15)2-3-8(7)12/h2-4,12H,1H3,(H,10,11)(H2,13,14,15)
		⚫	| SMILES1 = CC(=O)NC1=CC(=CC=C1O)(O)(O)=O
⚫	| StdInChI_Ref = {{stdinchicite|correct|chemspider}}
	| InChI = 1/C8H10AsNO5/c1-5(11)10-7-4-6(9(13,14)15)2-3-8(7)12/h2-4,12H,1H3,(H,10,11)(H2,13,14,15)		| StdInChI = 1S/C8H10AsNO5/c1-5(11)10-7-4-6(9(13,14)15)2-3-8(7)12/h2-4,12H,1H3,(H,10,11)(H2,13,14,15)
		⚫	| StdInChI_Ref = {{stdinchicite|correct|chemspider}}
⚫	| StdInChIKey = ODFJOVXVLFUVNQ-UHFFFAOYSA-N
		⚫	| InChI = 1/C8H10AsNO5/c1-5(11)10-7-4-6(9(13,14)15)2-3-8(7)12/h2-4,12H,1H3,(H,10,11)(H2,13,14,15)
⚫	| StdInChIKey_Ref = {{stdinchicite|correct|chemspider}}
	| InChIKey = ODFJOVXVLFUVNQ-UHFFFAOYAX}}		| StdInChIKey = ODFJOVXVLFUVNQ-UHFFFAOYSA-N
		⚫	| StdInChIKey_Ref = {{stdinchicite|correct|chemspider}}
⚫	| Section2 = {{Chembox Properties
		⚫	| InChIKey = ODFJOVXVLFUVNQ-UHFFFAOYAX}}
	| C = 8
		⚫	|Section2={{Chembox Properties
	| H = 10
	| As = 1		| C=8|As=1|N=1|H=10|O=5
		⚫	| MolarMass = 275.0903 g mol<sup>−1</sup>
	| N = 1
			}}
	| O = 5
			|Section6={{Chembox Pharmacology
⚫	| ExactMass = 274.977493852 g mol<sup>-1</sup>}}
		⚫	| ATCCode_prefix = A07
			| ATCCode_suffix = AX02
			| ATC_Supplemental = {{ATC|G01|AB01}}, {{ATC|P01|CD02}}, {{ATC|P51|AD05}}
			}}
			|Section7={{Chembox Hazards
			| GHSPictograms = {{GHS skull and crossbones}} {{GHS environment}}
			| GHSSignalWord = Danger
			| HPhrases = {{H-phrases|301|331|410}}
			| PPhrases = {{P-phrases|261|273|301+310|311|501}}
			}}
	}}		}}
⚫	'''Acetarsol''' is an anti-infective.<ref name="pmid12035784">{{cite journal |author=Chen MY, Smith NA, Fox EF, Bingham JS, Barlow D |title=Acetarsol pessaries in the treatment of metronidazole resistant Trichomonas vaginalis |journal=Int J STD AIDS |volume=10 |issue=4 |pages=277–80 |year=1999 |month=April |pmid=12035784 |doi= 10.1258/0956462991913943|url=http://ijsa.rsmjournals.com/cgi/pmidlookup?view=long&pmid=12035784}}</ref>
		⚫	'''Acetarsol''' (or '''acetarsone'''<ref>{{cite web|url=https://fdasis.nlm.nih.gov/srs/unii/806529YU1N|title=FDA Substance Registration System: Acetarsol|accessdate=6 May 2021|archive-date=8 January 2021|archive-url=https://web.archive.org/web/20210108134948/https://fdasis.nlm.nih.gov/srs/unii/806529yu1n|url-status=dead}}</ref>) is an anti-] drug.<ref name="pmid12035784">{{cite journal |vauthors=Chen MY, Smith NA, Fox EF, Bingham JS, Barlow D |title=Acetarsol pessaries in the treatment of metronidazole resistant Trichomonas vaginalis |journal=Int J STD AIDS |volume=10 |issue=4 |pages=277–80 |date=April 1999 |pmid=12035784 |doi= 10.1258/0956462991913943|s2cid=27353282 |url=http://ijsa.rsmjournals.com/cgi/pmidlookup?view=long&pmid=12035784}}</ref>
	It was first discovered in 1921 at ] by Ernest Fourneau ], and sold under the brand name '''Stovarsol''' (''fourneau'' is the French word for stove). <ref></ref> <ref>''Traité de chimie organique'', sous la direction de Victor Grignard, Paul Baud, vol. 22, Masson, 1959, p. 1127-1130.</ref>
	It has been given in ].<ref name="pmid15352902">{{cite journal |author=Gionchetti P, Rizzello F, Morselli C, Campieri M |title=Review article: problematic proctitis and distal colitis |journal=Aliment. Pharmacol. Ther. |volume=20 Suppl 4 |issue= |pages=93–6 |year=2004 |month=October |pmid=15352902 |doi=10.1111/j.1365-2036.2004.02049.x |url=http://www3.interscience.wiley.com/resolve/openurl?genre=article&sid=nlm:pubmed&issn=0269-2813&date=2004&volume=20&issue=&spage=93}}</ref>		It was first discovered in 1921 at ] by ],<ref name=":0">{{cite web|last=PubChem|title=Acetarsol|url=https://pubchem.ncbi.nlm.nih.gov/compound/1985|access-date=2021-03-31|website=pubchem.ncbi.nlm.nih.gov|language=en}}</ref> and sold under the brand name '''Stovarsol'''.<ref>{{cite web |url=http://www.ordre.pharmacien.fr/upload/Syntheses/161.pdf |title=Éric Fouassier, ''Ces poisons qui guérissent'', oct. 1996, p. 5. |access-date=2010-04-01 |archive-date=2011-10-05 |archive-url=https://web.archive.org/web/20111005185843/http://www.ordre.pharmacien.fr/upload/Syntheses/161.pdf |url-status=dead }}</ref><ref>''Traité de chimie organique'', sous la direction de Victor Grignard, Paul Baud, vol. 22, Masson, 1959, p. 1127-1130.</ref> It has been given in the form of ].<ref name="pmid15352902">{{cite journal |vauthors=Gionchetti P, Rizzello F, Morselli C, Campieri M |title=Review article: problematic proctitis and distal colitis |journal=Aliment. Pharmacol. Ther. |volume=20 |pages=93–6 |date=October 2004 |issue=Suppl 4 |pmid=15352902 |doi=10.1111/j.1365-2036.2004.02049.x |s2cid=72699260 |doi-access=free }}</ref>
			Acetarsol can be used to make ].{{cn|date=December 2022}}
			It has been cancelled and withdrawn from the market since August 12th, 1997.<ref name=":0" />
			== Medical uses ==
			Acetarsol has been used for the treatment of diseases such as ], ], ], trypanosomiasisiasis and ]. Acetarsol was used for the treatment of ''Trichomonas Vaginalis'' and ''Candida Albicans.'' In the oral form, acetarsol can be used for the treatment of ]. As a suppository, acetarsol was researched to be used for the treatment of proctitis.<ref name=":0" />
			== Mechanism of action ==
			Although the mechanism of action is not fully known, acetarsol may bind to protein-containing ] groups located in the parasite, which then creates lethal As-S bonds, which then kills the parasite. <ref name=":0" />
			== Chemistry and pharmacokinetics ==
			Acetarsol has the molecular formula ''N''-acetyl-4-hydroxy-''m''-arsinillic acid, and it is a ] ] compound with ] and ] properties. The arsenic found in acetarsol is excreted mainly in urine. The level of arsenic after acetarsol administration reaches close to the toxic range in urine.<ref name=":0" /> Some reports indicate a remission of arsenic which can be physiologically dangerous. <ref name=":0" />
			== Toxicity ==
			Some reports indicate that acetarsol can produce effects in the eyes such as optic ] and ].<ref>{{cite web|last=PubChem|title=Acetarsol|url=https://pubchem.ncbi.nlm.nih.gov/compound/1985|access-date=2022-01-16|website=pubchem.ncbi.nlm.nih.gov|language=en}}</ref>
	==References==		==References==
	{{reflist}}		{{Reflist}}
	{{Antidiarrheals, intestinal anti-inflammatory/anti-infective agents}}		{{Antidiarrheals, intestinal anti-inflammatory/anti-infective agents}}
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	]		]
	]		]
	]
	]		]
	{{gastrointestinal-drug-stub}}
	{{antiinfective-drug-stub}}
	{{genito-urinary-drug-stub}}
	]
	]
	]
	]