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{{short description|Derivative of aspartic acid found in the brain}} |
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{{ambox | text = This page contains a copy of the infobox ({{tl|chembox}}) taken from revid of page ] with values updated to verified values.}} |
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{{DISPLAYTITLE:''N''-Acetylaspartic acid}} |
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{{Chembox |
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{{chembox |
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| Verifiedfields = changed |
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| Verifiedfields = changed |
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| Watchedfields = changed |
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| Watchedfields = changed |
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| Name = ''N''-Acetylaspartic acid |
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| Name = ''N''-Acetylaspartic acid |
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| verifiedrevid = 462256723 |
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| verifiedrevid = 477506883 |
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| ImageFile = Acetylaspartate.png |
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| ImageFile = Acetylaspartate.png |
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| ImageFile_Ref = {{chemboximage|correct|??}} |
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| ImageFile_Ref = {{chemboximage|correct|??}} |
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| ImageSize = 160 |
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| ImageName = Stereo, skeletal formula of N-acetylaspartic acid (S) |
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| ImageName = Stereo, skeletal formula of N-acetylaspartic acid (S) |
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| IUPACName = 2-Acetamidobutanedioic acid<ref>{{Cite web|title=N-acetylaspartate - Compound Summary|url=http://pubchem.ncbi.nlm.nih.gov/summary/summary.cgi?cid=97508|work=PubChem Compound|publisher=National Center for Biotechnology Information|accessdate=8 January 2012|location=USA|date=26 March 2005|at=Identification and Related Records}}</ref> |
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| IUPACName = 2-Acetamidobutanedioic acid<ref>{{cite web|title=N-acetylaspartate - Compound Summary|url=https://pubchem.ncbi.nlm.nih.gov/summary/summary.cgi?cid=97508|work=PubChem Compound|publisher=National Center for Biotechnology Information|access-date=8 January 2012|location=USA|date=26 March 2005|at=Identification}}</ref> |
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|Section1={{Chembox Identifiers |
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| OtherNames = {{Unbulleted list|''N''-Acetylaspartate{{Citation needed|date=January 2012}}|Acetylaspartic acid{{Citation needed|date=January 2012}} |
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| CASNo = 2545-40-6 |
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| UNII_Ref = {{fdacite|correct|FDA}} |
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| UNII = 445Y04YIWR |
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| CASNo_Ref = {{cascite|correct|CAS}} |
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| CASNo1 = 997-55-7 |
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| CASNo1_Ref = {{cascite|correct|CAS}} |
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| CASNo1_Comment = <small>''S''</small> |
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| PubChem = 97508 |
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| PubChem1 = 774916 |
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| PubChem1_Comment = <small>''R''</small> |
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| PubChem2 = 65065 |
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| PubChem2_Comment = <small>''S''</small> |
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| ChemSpiderID = 88007 |
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| ChemSpiderID_Ref = {{chemspidercite|changed|chemspider}} |
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| ChemSpiderID1 = 677387 |
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| ChemSpiderID1_Ref = {{chemspidercite|correct|chemspider}} |
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| ChemSpiderID1_Comment = <small>''R''</small> |
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| EINECS = 219-827-5 |
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| KEGG = C01042 |
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| KEGG_Ref = {{keggcite|changed|kegg}} |
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| MeSHName = N-acetylaspartate |
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| ChEBI = 21547 |
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| ChEBI_Ref = {{ebicite|correct|EBI}} |
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| ChEMBL = 1162493 |
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| ChEMBL_Ref = {{ebicite|changed|EBI}} |
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| RTECS = CI9098600 |
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| Beilstein = 1726198 <small>''S''</small> |
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| 3DMet = B00227 |
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| SMILES = CC(=O)N(CC(=O)O)C(=O)O |
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| StdInChI = 1S/C6H9NO5/c1-3(8)7-4(6(11)12)2-5(9)10/h4H,2H2,1H3,(H,7,8)(H,9,10)(H,11,12) |
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| StdInChI_Ref = {{stdinchicite|changed|chemspider}} |
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| StdInChIKey = OTCCIMWXFLJLIA-UHFFFAOYSA-N |
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| StdInChIKey_Ref = {{stdinchicite|changed|chemspider}} |
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}} |
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}} |
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| Section1 = {{Chembox Identifiers |
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|Section2={{Chembox Properties |
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| C=6 | H=9 | N=1 | O=5 |
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| Abbreviations = NAA{{Citation needed|date=January 2012}} |
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| Appearance = Colourless, transparent crystals |
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| CASNo = 997-55-7 |
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| MeltingPtC = 137 to 140 |
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| CASNo_Ref = {{cascite|changed|??}} |
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| BoilingPtC = 141 to 144 |
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| CASNo1 = 997-55-7 |
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| LogP = −2.209 |
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| CASNo1_Ref = {{cascite|correct|CAS}} |
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| pKa = 3.142 |
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| CASNo1_Comment = <small>(''S'')</small> |
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| PubChem = 97508 |
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| pKb = 10.855 |
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| PubChem_Ref = {{Pubchemcite|correct|Pubchem}} |
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| PubChem1 = 774916 |
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| PubChem1_Ref = {{Pubchemcite|correct|Pubchem}} |
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| PubChem1_Comment = <small>(''R'')</small> |
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| PubChem2 = 65065 |
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| PubChem2_Ref = {{Pubchemcite|correct|Pubchem}} |
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| PubChem2_Comment = <small>(''S'')</small> |
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| ChemSpiderID = 58576 |
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| ChemSpiderID_Ref = {{chemspidercite|changed|chemspider}} |
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| ChemSpiderID1 = 677387 |
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| ChemSpiderID1_Ref = {{chemspidercite|correct|chemspider}} |
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| ChemSpiderID1_Comment = <small>(''R'')</small> |
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| EINECS = 219-827-5 |
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| KEGG = <!-- blanked - oldvalue: C01042 --> |
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| KEGG_Ref = {{keggcite|changed|kegg}} |
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| MeSHName = N-acetylaspartate |
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| ChEBI = 21547 |
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| ChEBI_Ref = {{ebicite|correct|EBI}} |
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| ChEMBL = 1162494 |
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| ChEMBL_Ref = {{ebicite|changed|EBI}} |
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| RTECS = CI9098600 |
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| Beilstein = 1726198 <small>(''S'')</small> |
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| 3DMet = B00227 |
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| SMILES = CC(=O)NC(CC(O)=O)C(O)=O |
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| StdInChI = 1S/C6H9NO5/c1-3(8)7-4(6(11)12)2-5(9)10/h4H,2H2,1H3,(H,7,8)(H,9,10)(H,11,12)/t4-/m0/s1 |
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| StdInChI_Ref = {{stdinchicite|changed|chemspider}} |
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| StdInChIKey = OTCCIMWXFLJLIA-BYPYZUCNSA-N |
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| StdInChIKey_Ref = {{stdinchicite|changed|chemspider}} |
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}} |
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}} |
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| Section2 = {{Chembox Properties |
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|Section3={{Chembox Hazards |
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| GHSPictograms = {{GHS07}} |
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| C=6|H=9|N=1|O=5 |
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| GHSSignalWord = Warning |
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| ExactMass = 175.048072403 g mol<sup>1−</sup> |
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| HPhrases = {{H-phrases|315|319|335}} |
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| Appearance = Colourless, transparent crystals |
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| PPhrases = {{P-phrases|261|264|271|280|302+352|304+340|305+351+338|312|321|332+313|337+313|362|403+233|405|501}} |
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| MeltingPtCL = 137 |
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| MeltingPtCH = 140 |
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| BoilingPtCL = 141 |
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| BoilingPtCH = 144 |
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| LogP = −2.209 |
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| pKa = 3.142 |
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| pKb = 10.855 |
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}} |
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}} |
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| Section3 = {{Chembox Hazards |
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|Section4={{Chembox Related |
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| OtherFunction_label = alkanoic acids |
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| SPhrases = {{S22}}, {{S24/25}} |
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| OtherFunction = {{unbulleted list|]|]|]|]|]|]}} |
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}} |
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| OtherCompounds = {{unbulleted list|]|]}} |
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| Section4 = {{Chembox Related |
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| OtherCpds = ] |
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}} |
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}} |
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}} |
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}} |
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'''''N''-Acetylaspartic acid''', or '''''N''-acetylaspartate''' ('''NAA'''), is a derivative of ] with a formula of C<sub>6</sub>H<sub>9</sub>NO<sub>5</sub> and a molecular weight of 175.139. |
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NAA is the second-most-concentrated ] in the ] after the ] ]. It is detected in the adult brain in ]s,<ref>{{cite journal | vauthors = Simmons ML, Frondoza CG, Coyle JT | title = Immunocytochemical localization of N-acetyl-aspartate with monoclonal antibodies | journal = Neuroscience | volume = 45 | issue = 1 | pages = 37–45 | date = 1991 | pmid = 1754068 | doi = 10.1016/0306-4522(91)90101-s | s2cid = 24071454 }}</ref> ]s and ]<ref name="ReferenceA">{{cite journal | vauthors = Nordengen K, Heuser C, Rinholm JE, Matalon R, Gundersen V | title = Localisation of N-acetylaspartate in oligodendrocytes/myelin | journal = Brain Structure & Function | volume = 220 | issue = 2 | pages = 899–917 | date = March 2015 | pmid = 24379086 | doi = 10.1007/s00429-013-0691-7 | s2cid = 475973 }}</ref> and is synthesized in the ] from the amino acid ] and ].<ref>{{cite journal | vauthors = Patel TB, Clark JB | title = Synthesis of N-acetyl-L-aspartate by rat brain mitochondria and its involvement in mitochondrial/cytosolic carbon transport | journal = The Biochemical Journal | volume = 184 | issue = 3 | pages = 539–46 | date = December 1979 | doi = 10.1042/bj1840539 | pmid = 540047 | pmc = 1161835 }}</ref> |
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== Function == |
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The various functions served by NAA are under investigation, but the primary proposed functions include: |
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* Neuronal ] that is involved in fluid balance in the brain |
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* Source of ] for ] and myelin synthesis in oligodendrocytes, the ] cells that myelinate neuronal axons |
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* Precursor for the synthesis of the neuronal dipeptide ] |
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* Contributor to energy production from the amino acid ] in neuronal mitochondria |
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In the brain, NAA was thought to be present predominantly in neuronal cell bodies, where it acts as a neuronal marker,<ref name="PMD11406719">{{cite journal | vauthors = Chatham JC, Blackband SJ | title = Nuclear magnetic resonance spectroscopy and imaging in animal research | journal = ILAR Journal | volume = 42 | issue = 3 | pages = 189–208 | year = 2001 | pmid = 11406719 | doi = 10.1093/ilar.42.3.189 | doi-access = free }}</ref> but it is also free to diffuse throughout neuronal fibers.<ref>{{cite journal | vauthors = Najac C, Branzoli F, Ronen I, Valette J | title = Brain intracellular metabolites are freely diffusing along cell fibers in grey and white matter, as measured by diffusion-weighted MR spectroscopy in the human brain at 7 T | journal = Brain Structure & Function | volume = 221 | issue = 3 | pages = 1245–54 | date = April 2016 | pmid = 25520054 | pmc = 4878649 | doi = 10.1007/s00429-014-0968-5 }}</ref> |
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== Applications == |
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However, the recent discovery of a higher concentration of NAA in myelin and oligodendrocytes than in neurons raises questions about the validity of the use of NAA as a neuronal marker.<ref name="ReferenceA" /> NAA gives off the largest signal in ] of the human brain. The levels measured there are decreased in numerous neuropathological conditions ranging from brain injury to ] to ]. This fact makes NAA a potential diagnostic molecule for doctors treating patients with brain damage or disease. |
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NAA may be a marker of creativity.<ref>{{cite web|url=https://www.newscientist.com/article/mg20227084.300-creativity-chemical-favours-the-smart.html|title=Creativity chemical favours the smart|first=Linda|last=Geddes}}</ref> High NAA levels in the ] are related to better ] performance in humans.<ref>{{cite journal | vauthors = Kozlovskiy S, Vartanov A, Pyasik M, Polikanova I | year = 2012 | title = Working memory and N-acetylaspartate level in hippocampus, parietal cortex and subventricular zone | journal = International Journal of Psychology | volume = 47 | page = 584 | doi = 10.1080/00207594.2012.709117 | doi-access = free }}</ref> Whole-brain levels of NAA have also been found to be positively correlated with educational attainment in adults.<ref> |
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{{cite journal |
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| date = 30 October 2012 |
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| title = The whole-brain N-acetylaspartate correlates with education in normal adults |
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| url = https://doi.org/10.1016%2Fj.pscychresns.2012.04.013 |
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| vauthors = Glodzik L, Wu WE, Babb JS, Achtnichts L, Amann M, Sollberger M, Monsch AU, Gass A, Gonenb O |
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| journal = Psychiatry Research: Neuroimaging |
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| volume = 204 |
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| issue = 1 |
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| pages = 49–54 |
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| doi = 10.1016/j.pscychresns.2012.04.013 |
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| pmid = 23177924 |
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| access-date = |
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| pmc = 3508436 |
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}} |
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</ref> |
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NAA may function as a ] in the brain by acting on ]s.<ref name="pmid12919386">{{cite journal | vauthors = Yan HD, Ishihara K, Serikawa T, Sasa M | title = Activation by N-acetyl-L-aspartate of acutely dissociated hippocampal neurons in rats via metabotropic glutamate receptors | journal = Epilepsia | volume = 44 | issue = 9 | pages = 1153–9 | date = September 2003 | pmid = 12919386 | doi = 10.1046/j.1528-1157.2003.49402.x | s2cid = 39902618 | doi-access = free }}</ref> |
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== See also == |
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* ] |
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* ] |
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== References == |
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{{reflist|32em}} |
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== Further reading == |
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{{refbegin}} |
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* {{cite book|editor-first1=John |editor-last1=Moffett|editor-first2=Suzannah B.|editor-last2= Tieman|editor-first3=Daniel R. |editor-last3=Weinberger|editor-first4=Joseph T. |editor-last4=Coyle |editor-first5=Aryan M. A. |editor-last5=Namboodiri | name-list-style = vanc |title=N-Acetylaspartate: A Unique Neuronal Molecule in the Central Nervous System|url={{google books |plainurl=y |id=tR44q6WWRBgC}}|date=21 October 2006|publisher=Springer Science & Business Media|isbn=978-0-387-30172-3}} |
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*{{cite journal | vauthors = Jung RE, Gasparovic C, Chavez RS, Flores RA, Smith SM, Caprihan A, Yeo RA | title = Biochemical support for the "threshold" theory of creativity: a magnetic resonance spectroscopy study | journal = The Journal of Neuroscience | volume = 29 | issue = 16 | pages = 5319–25 | date = April 2009 | pmid = 19386928 | pmc = 2755552 | doi = 10.1523/JNEUROSCI.0588-09.2009 }} |
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{{refend}} |
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== External links == |
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* |
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{{Neurotransmitters}} |
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{{Glutamatergics}} |
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{{DEFAULTSORT:Acetylaspartic acid, N-}} |
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] |
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] |
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] |